Synthesis, physico-chemical properties and antimicrobial activity of novel 4-arylamino-2-methylquinolines
Keywords:
4-arylaminoquinolines, 4-chloroqumolines, antimicrobial activity
Abstract
Synthesis of novel 4-arylaminoquinolines has been carried out, its physico-chemical characteristics and antimicrobial activity has been studied. It has been shown that new 4-arylaminoquinolines have moderate levels of antimicrobial and antifungal activity. QSAR analisys has been carried out for these derivatives.
References
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6. Casagrande M., Basilico N., Parapini S. et al. // Bioorg. and Med. Chem.— 2008, Vol. 16, No. 14. P. 6813-6823.
7. Solomon V.R., Puri S.K., Srivastava K. et al. // Ibid. - 2005. - Vol. 13, 6. P. 2157-2165.
8. Sparatore A., Basilico N., Casagrande M. et al. // Bioorg. and Med. Chem. Letters. - 2008, - Vol. 18, No. 13. P. 3737-3740.
Published
2020-07-09
How to Cite
Gritsenko, I., Zubkov, V., & Podolsky, I. (2020). Synthesis, physico-chemical properties and antimicrobial activity of novel 4-arylamino-2-methylquinolines. Farmatsevtychnyi Zhurnal, (5), 70-75. Retrieved from https://pharmj.org.ua/index.php/journal/article/view/917
Section
Original Articles
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